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产品介绍 PDE InhibitorOur Inhibitors are extremely Pure
询价产品介绍 PDE Inhibitor
询价产品介绍 PRMT1,3,4 &6 Inhibitor
询价产品介绍 UNC0321 (trifluoroacetate salt) is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP (also known as EHMT1), with IC50 of 6 nM and 15 nM, respectively. It is more than 40,000-fold more selective for G9a and GLP vs. SET7/9, SET8, PRMT3, or JMJD2E.
询价产品介绍 Tranylcypromine (2-PCPA) is an irreversible inhibitor of LSD1 histone demethylase and monoamine oxidases (MAO). The inhibitor targets monoamine oxidases A and B and has been used as a chemical scaffold to design new demethylase inhibitors. Tranylcypromine has been shown to increase Histone H3 lysine 4 (H3K4) methylation in P19 embryonal carcinoma cell.
询价产品介绍 UNC0224 is a potent and selective inhibitor of G9a, a histone methyltransferase (HMT). It also inhibits GLP, a closely-related H3K9 HMT, but is more than 1,000-fold selective against SET7/9 and SET8.
询价产品介绍 CP 80633 is a selective inhibitor of PDE4, which does not display significant isozyme selectivity. It also inhibits hydrolysis of cAMP in isolated monocytes, eosinophils, human peripheral blood and T-cells. It has been shown to exhibit anti-inflammatory and bronchodilatory activity in vivo.
询价产品介绍 Aliskiren Hydrochloride is an orally active, synthetic nonpeptide Renin inhibitor that has been shown to work as an antihypertensive.
询价产品介绍 (S)-MG132, also known as Z-Leu-Leu-Leu-CHO, is a potent, reversible and cell-permeable inhibitor of proteasomes that inhibits cell growth in B16 and IPC227F cells. It also inhibits NF-κB activation, sensitizing a variety of carcinoma cell lines to apoptosis.
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